CMap Candidate Details
Structure:
| CMap ID: | C02430 |
| Pert ID: | BRD-K60341624 |
| Compound Name: | GSK1292263 |
| Targets: | GRPR |
| MoA: | glucose dependent insulinotropic receptor agonist |
| SMILES: | CC(C)c1noc(n1)N1CCC(COc2ccc(nc2)-c2ccc(cc2)S(C)(=O)=O)CC1 |
| InchiKey: | |
| Compound Aliases: |
| Score ID | Pert ID | Cell Line | Pert Dose | Pert Time | Raw Score (GSE126848) | Normalized Score (GSE126848) | fdr_q_nlog10 (GSE126848) | Raw Score (GSE135251) | Normalized Score (GSE135251) | fdr_q_nlog10 (GSE135251) |
|---|---|---|---|---|---|---|---|---|---|---|
| 123538 | BRD-K60341624 | HA1E | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.37 | -1.26 | 1.35 |
| 123573 | BRD-K60341624 | HEK293 | 1.11 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.38 | -1.27 | 1.39 |
| 123649 | BRD-K60341624 | HT29 | 10 uM | 24 h | 0.27 | 1.11 | 0.25 | 0.27 | 0.97 | 0.35 |
| 123690 | BRD-K60341624 | MCF10A | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.3 | -1.01 | 0.56 |
| 123766 | BRD-K60341624 | YAPC | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.22 | -0.73 | 0.04 |
| 131981 | BRD-K60341624 | A375 | 2.22 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.34 | -1.16 | 1.11 |
| 132036 | BRD-K60341624 | HELA | 0.74 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 132081 | BRD-K60341624 | MCF??7.00 | 2.22 uM | 24 h | -0.28 | -1.18 | 0.5 | 0.0 | 0.0 | 0.0 |
| 132113 | BRD-K60341624 | PC3 | 2.22 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |