CMap Candidate Details
Structure:
| CMap ID: | C01532 |
| Pert ID: | BRD-K22482860 |
| Compound Name: | dalfampridine |
| Targets: | KCNA1|KCNA10|KCNA2|KCNA3|KCNA4|KCNA5|KCNA6|KCNA7|KCNB1|KCNB2|KCNC1|KCNC2|KCNC3|KCNC4|KCND1|KCND2|KCND3|KCNF1|KCNG1|KCNG2|KCNG3|KCNG4|KCNH1|KCNH2|KCNH3|KCNH4|KCNH5|KCNH6|KCNH7|KCNH8|KCNJ13|KCNJ5|KCNQ1|KCNQ2|KCNQ3|KCNQ4|KCNQ5|KCNS1|KCNS2|KCNS3|KCNV1|KCNV2 |
| MoA: | potassium channel blocker |
| SMILES: | Nc1ccncc1 |
| InchiKey: | |
| Compound Aliases: |
| Score ID | Pert ID | Cell Line | Pert Dose | Pert Time | Raw Score (GSE126848) | Normalized Score (GSE126848) | fdr_q_nlog10 (GSE126848) | Raw Score (GSE135251) | Normalized Score (GSE135251) | fdr_q_nlog10 (GSE135251) |
|---|---|---|---|---|---|---|---|---|---|---|
| 121373 | BRD-K22482860 | A375 | 1.11 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 121389 | BRD-K22482860 | HA1E | 3.33 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 121419 | BRD-K22482860 | HELA | 0.125 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.2 | -0.69 | 0.02 |
| 121468 | BRD-K22482860 | MCF??7.00 | 0.125 uM | 24 h | 0.19 | 0.79 | 0.0 | 0.0 | 0.0 | 0.0 |
| 121531 | BRD-K22482860 | YAPC | 0.04 uM | 24 h | 0.24 | 0.99 | 0.09 | 0.0 | 0.0 | 0.0 |
| 129500 | BRD-K22482860 | HT29 | 0.01 uM | 24 h | -0.3 | -1.26 | 0.71 | -0.33 | -1.1 | 0.87 |
| 129564 | BRD-K22482860 | PC3 | 0.08 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |