CMap Candidate Details
Structure:
| CMap ID: | C03543 |
| Pert ID: | BRD-K94853001 |
| Compound Name: | Mps1-IN-1 |
| Targets: | TTK |
| MoA: | monopolar spindle 1 kinase inhibitor |
| SMILES: | COc1cc(ccc1Nc1cc(Nc2ccccc2S(=O)(=O)C(C)C)c2cc[nH]c2n1)N1CCC(O)CC1 |
| InchiKey: | |
| Compound Aliases: |
| Score ID | Pert ID | Cell Line | Pert Dose | Pert Time | Raw Score (GSE126848) | Normalized Score (GSE126848) | fdr_q_nlog10 (GSE126848) | Raw Score (GSE135251) | Normalized Score (GSE135251) | fdr_q_nlog10 (GSE135251) |
|---|---|---|---|---|---|---|---|---|---|---|
| 50 | BRD-K94853001 | BJAB | 10 uM | 4 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 84 | BRD-K94853001 | HBL1 | 0.66 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.3 | 1.05 | 0.57 |
| 120 | BRD-K94853001 | K562 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 172 | BRD-K94853001 | KMS34 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.26 | -0.86 | 0.21 |
| 214 | BRD-K94853001 | NALM6 | 0.125 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 253 | BRD-K94853001 | OCILY10 | 0.01 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 284 | BRD-K94853001 | OCILY19 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 349 | BRD-K94853001 | OCILY3 | 10 uM | 4 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 370 | BRD-K94853001 | SKMEL5 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.25 | 0.89 | 0.21 |
| 419 | BRD-K94853001 | THP1 | 10 uM | 4 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 440 | BRD-K94853001 | TMD8 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.27 | -0.92 | 0.34 |