CMap Candidate Details
Structure:
| CMap ID: | C04397 |
| Pert ID: | BRD-K75089421 |
| Compound Name: | procainamide |
| Targets: | DNMT1|SCN5A |
| MoA: | sodium channel blocker |
| SMILES: | CCN(CC)CCNC(=O)c1ccc(N)cc1 |
| InchiKey: | |
| Compound Aliases: |
| Score ID | Pert ID | Cell Line | Pert Dose | Pert Time | Raw Score (GSE126848) | Normalized Score (GSE126848) | fdr_q_nlog10 (GSE126848) | Raw Score (GSE135251) | Normalized Score (GSE135251) | fdr_q_nlog10 (GSE135251) |
|---|---|---|---|---|---|---|---|---|---|---|
| 4483 | BRD-K75089421 | HCC515 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 37732 | BRD-K75089421 | ASC | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.35 | -1.17 | 1.12 |
| 38549 | BRD-K75089421 | NPC | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.33 | -1.11 | 0.92 |
| 38773 | BRD-K75089421 | PHH | 10 uM | 24 h | 0.23 | 0.97 | 0.08 | 0.25 | 0.89 | 0.2 |
| 51178 | BRD-K75089421 | VCAP | 10 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 90983 | BRD-K75089421 | HUH7 | 15 uM | 72 h | 0.0 | 0.0 | 0.0 | -0.24 | -0.82 | 0.15 |
| 127016 | BRD-K75089421 | A375 | 3.33 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 127095 | BRD-K75089421 | HELA | 0.04 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.19 | -0.63 | 0.0 |
| 127136 | BRD-K75089421 | HT29 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 127163 | BRD-K75089421 | JURKAT | 0.37 uM | 24 h | -0.22 | -0.91 | 0.06 | -0.43 | -1.45 | 15.35 |
| 127206 | BRD-K75089421 | MCF??7.00 | 0.37 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 127235 | BRD-K75089421 | PC3 | 0.125 uM | 24 h | -0.2 | -0.83 | 0.0 | -0.25 | -0.85 | 0.19 |
| 127278 | BRD-K75089421 | THP1 | 0.37 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.28 | 1.0 | 0.43 |
| 127309 | BRD-K75089421 | YAPC | 0.125 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 135040 | BRD-K75089421 | A549 | 2.22 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 135082 | BRD-K75089421 | HA1E | 0.01 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 135106 | BRD-K75089421 | HEK293 | 0.08 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.26 | -0.89 | 0.26 |
| 135203 | BRD-K75089421 | MCF10A | 0.08 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 135259 | BRD-K75089421 | MDAMB231 | 0.74 uM | 24 h | 0.26 | 1.08 | 0.22 | 0.0 | 0.0 | 0.0 |