Bioactive Compound Details
| Compound ID: | B1380102 |
| Source ID: | CHEMBL2107832 |
| Source Type: | Small molecule |
| Compound Name: | PIMASERTIB |
| Synonyms: | AS 703026|As-703026|AS-703026|AS703026|EMD 1036239|EMD-1036239|G-02443714|Msc-1936369|MSC-1936369A|MSC-1936369B|MSC1936369A|Msc1936369a; as703026; emd 1036239|Pimasertib|Pimasertib|Pimasertib |
| Molecular Formula: | C15H15FIN3O3 |
| SMILES: | O=C(NC[C@H](O)CO)c1ccncc1Nc1ccc(I)cc1F |
| Molecular Species: | NEUTRAL |
| Target ID | Target Name | GENE | Action | Class | UniProtKB ID | Entry Name | |
|---|---|---|---|---|---|---|---|
| T09 | Serine/threonine-protein kinase AKT2 | AKT2 | INHIBITOR | Target is a single protein chain | P31751 | AKT2_HUMAN | Details |
| T09 | Serine/threonine-protein kinase AKT2 | AKT2 | INHIBITOR | Target is a single protein chain | P31751 | AKT2_HUMAN | Details |
| T30 | TP53-regulating kinase | TP53RK | Target is a single protein chain | Q96S44 | TP53RK_HUMAN | Details | |
| T01 | Insulin receptor | INSR | AGONIST; INHIBITOR | Target is a single protein chain | P06213 | INSR_HUMAN | Details |