Bioactive Compound Details
| Compound ID: | B1675825 |
| Source ID: | CHEMBL3186534 |
| Source Type: | Small molecule |
| Compound Name: | RIVOCERANIB |
| Synonyms: | Apatinib|Apatinib free base|Rivoceranib|Rivoceranib|Rivoceranib|YN968D1|YN968D1 FREE BASE |
| Molecular Formula: | C24H23N5O |
| SMILES: | N#CC1(c2ccc(NC(=O)c3cccnc3NCc3ccncc3)cc2)CCCC1 |
| Molecular Species: | NEUTRAL |
| Target ID | Target Name | GENE | Action | Class | UniProtKB ID | Entry Name | |
|---|---|---|---|---|---|---|---|
| T09 | Serine/threonine-protein kinase AKT2 | AKT2 | INHIBITOR | Target is a single protein chain | P31751 | AKT2_HUMAN | Details |
| T09 | Serine/threonine-protein kinase AKT2 | AKT2 | INHIBITOR | Target is a single protein chain | P31751 | AKT2_HUMAN | Details |
| T30 | TP53-regulating kinase | TP53RK | Target is a single protein chain | Q96S44 | TP53RK_HUMAN | Details | |
| T01 | Insulin receptor | INSR | AGONIST; INHIBITOR | Target is a single protein chain | P06213 | INSR_HUMAN | Details |