CMap Candidates
CMap (Connectivity Map) candidates are extracted from CLUE (CMap and LINCS Unified Environment), with detailed information, e.g., perturbagen time and dose, compound structure, targets, SMILES, mechanism of action. Two publicly available gene expression profiles of CKD are used to calculate individual connectivity scores and corresponding statistical significances for these candidates.
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6125 records.
| CMap ID | Pert ID | Compound Name | Targets | MoA | Compound Aliases | |
|---|---|---|---|---|---|---|
| C04701 | BRD-K08640512 | RS-100329 | ADRA1A|ADRA1D | adrenergic receptor antagonist | Details | |
| C04702 | BRD-K87048468 | RS-102221 | HTR2A|HTR2B|HTR2C | serotonin receptor antagonist | Details | |
| C04703 | BRD-K83063356 | RS-102895 | CCR2 | CCR antagonist | Details | |
| C04704 | BRD-K90825648 | RS-127445 | HTR2A|HTR2B|HTR2C | serotonin receptor antagonist | Details | |
| C04705 | BRD-K80725821 | RS-16566 | serotonin receptor antagonist | Details | ||
| C04706 | BRD-K76840893 | RS-17053 | ADRA1A|ADRA1D | adrenergic receptor antagonist | Details | |
| C04707 | BRD-K01868942 | RS-23597-190 | HTR4 | serotonin receptor antagonist | Details | |
| C04708 | BRD-K20742498 | RS-39604 | HTR4 | serotonin receptor antagonist | Details | |
| C04709 | BRD-K26160755 | RS-45041-190 | imidazoline receptor agonist | Details | ||
| C04710 | BRD-K87510569 | RS-504393 | CCL2|CCR2 | CC chemokine receptor antagonist | Details | |
| C04711 | BRD-K20714604 | RS-56812 | HTR3A | serotonin receptor partial agonist | Details | |
| C04712 | BRD-K46142322 | RS-67333 | HTR4 | serotonin receptor partial agonist | Details | |
| C04713 | BRD-K50018155 | RS-67506 | HTR4 | serotonin receptor partial agonist | Details | |
| C04714 | BRD-K86600316 | RS-79948 | ADRA2A | adrenergic receptor antagonist | Details | |
| C04715 | BRD-K30159788 | RSV604 | RSV replication inhibitor | Details | ||
| C04716 | BRD-K56211775 | RTA-408 | NFE2L2 | nitric oxide production inhibitor | Details | |
| C04717 | BRD-A33603104 | RU-SKI-43 | HHAT | hedgehog pathway inhibitor | Details | |
| C04718 | BRD-K00234327 | RU-24969 | HTR1A|HTR1B|HTR1D|HTR2A|HTR2B|HTR2C|HTR5A|HTR6 | serotonin receptor agonist | Details | |
| C04719 | BRD-K37687387 | RU-28318 | NR3C2 | cytochrome P450 inhibitor | Details | |
| C04720 | BRD-K85285268 | RU-42173 | ADRB2 | adrenergic receptor agonist | Details | |
| C04721 | BRD-K62762455 | RU-58841 | AR | androgen receptor antagonist | Details | |
| C04722 | BRD-K79821389 | rubitecan | TOP1 | topoisomerase inhibitor | Details | |
| C04723 | BRD-K88560311 | rucaparib | PARP1|PARP2 | PARP inhibitor | Details | |
| C04724 | BRD-K61036791 | rucinol | TYR | tyrosinase inhibitor | Details | |
| C04725 | BRD-K20079257 | rufinamide | GRM5|SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A | voltage-gated sodium channel blocker | Details | |
| C04726 | BRD-K62374253 | rufloxacin | bacterial DNA gyrase inhibitor | Details | ||
| C04727 | BRD-K98004573 | rupatadine | HRH1|PTAFR | histamine receptor antagonist; platelet activating factor receptor antagonist | Details | |
| C04728 | BRD-K94723713 | rutaecarpine | PTGS2 | cyclooxygenase inhibitor | Details | |
| C04729 | BRD-K20482099 | rutin | AKR1C3 | antioxidant; capillary stabilizing agent; nitric oxide scavenger | Details | |
| C04730 | BRD-K53972329 | ruxolitinib | JAK1|JAK2|JAK3|TYK2 | JAK inhibitor | Details | |
| C04731 | BRD-K19601669 | ruxolitinib-(S) | JAK1|JAK2 | JAK inhibitor | Details | |
| C04732 | BRD-K00091711 | RWJ-21757 | TLR7 | toll-like receptor agonist | Details | |
| C04733 | BRD-K94623186 | RWJ-50271 | ICAM1 | integrin inhibitor | Details | |
| C04734 | BRD-K07074923 | RWJ-67657 | MAPK14|PTGS2 | MAP kinase inhibitor | Details | |
| C04735 | BRD-K66213167 | RX-3117 | CDK2|DNMT1 | DNA synthesis inhibitor; CDK inhibitor | Details | |
| C04736 | BRD-A65597028 | RX-821002 | ADRA1A|ADRA1B|ADRA1D|ADRA2A|ADRA2B|ADRA2C | adrenergic receptor antagonist | Details | |
| C04737 | BRD-K06426971 | ryuvidine | CDK2|CDK4 | histone lysine methyltransferase inhibitor | Details | |
| C04738 | BRD-K23902832 | R112 | SYK | syk inhibitor | Details | |
| C04739 | BRD-K86687746 | R306465 | HDAC inhibitor | Details | ||
| C04740 | BRD-K20285085 | R406 | RET|SYK | SYK inhibitor | Details | |
| C04741 | BRD-K52233191 | R547 | CDK1|CDK2|CDK4|CDK7 | CDK inhibitor | Details | |
| C04742 | BRD-K10673031 | S-Isopropylisothiourea | NOS3 | nitric oxide synthase inhibitor | Details | |
| C04743 | BRD-K63123526 | S-methylcysteine | CTSD|MGMT | Details | ||
| C04744 | BRD-K94780074 | S-Nitrosoglutathione | PTPN1 | nitric oxide stimulant | Details | |
| C04745 | BRD-K59527975 | S-Sulfo-L-cysteine-sodium-salt | glutamate receptor agonist | Details | ||
| C04746 | BRD-K09774593 | S-Trityl-L-cysteine | mitotic kinesin inhibitor | Details | ||
| C04747 | BRD-K37635256 | S-07662 | NR1I3 | CAR antagonist | Details | |
| C04748 | BRD-K60005752 | S-111 | PARP1 | PARP inhibitor | Details | |
| C04749 | BRD-K46766488 | S-14506 | HTR1A | serotonin receptor agonist | Details | |
| C04750 | BRD-K99819791 | SA-47 | FAAH | FAAH inhibitor | Details | |
| C04751 | BRD-K46493214 | saccharin | CA1|CA12|CA2|CA9 | DNA polymerase inhibitor | Details | |
| C04752 | BRD-A24122750 | saclofen | GABBR1|GABBR2|KCTD12|KCTD16|KCTD8 | GABA receptor antagonist | Details | |
| C04753 | BRD-K91456750 | sacubitril | MME | neprilysin inhibitor | Details | |
| C04754 | BRD-A96503329 | safflower-yellow | anti-inflammatory agent | Details | ||
| C04755 | BRD-K92613113 | safinamide | MAOB | dopamine uptake inhibitor; glutamate inhibitor; monoamine oxidase inhibitor | Details | |
| C04756 | BRD-K93944989 | safingol | TRPM3 | PKC inhibitor | Details | |
| C04757 | BRD-K90582192 | safranal | GABBR1 | benzodiazepine receptor agonist | Details | |
| C04758 | BRD-K99433989 | SAG | SMO|TRPC6 | smoothened receptor agonist | Details | |
| C04759 | BRD-K15045219 | salazodine | Details | |||
| C04760 | BRD-K64614248 | salicin | anti-inflammatory agent | Details | ||
| C04761 | BRD-K08493205 | salicyl-alcohol | Details | |||
| C04762 | BRD-K81130846 | salicylamide | analgesic agent | Details | ||
| C04763 | BRD-K83036479 | salicylanilide | other antibiotic | Details | ||
| C04764 | BRD-K93632104 | salicylic-acid | AKR1C1|PTGS1|PTGS2 | cyclooxygenase inhibitor | Details | |
| C04765 | BRD-K66030860 | salidroside | APP | beta amyloid protein neurotoxicity inhibitor | Details | |
| C04766 | BRD-A28301258 | salinomycin | Details | |||
| C04767 | BRD-K98453471 | salirasib | TRPA1 | mTOR inhibitor | Details | |
| C04768 | BRD-A01320529 | salmeterol | ADRB2 | adrenergic receptor agonist | Details | |
| C04769 | BRD-A49952467 | salsolinol-1-carboxylic-acid | Details | |||
| C04770 | BRD-A45107007 | salubrinal | EIF2S1 | eukaryotic translation initiation factor inhibitor | Details | |
| C04771 | BRD-K18898553 | salvianolic-acid-B | MMP9 | metalloproteinase inhibitor; EGFR inhibitor | Details | |
| C04772 | BRD-K19284129 | salvinorin-a | OPRD1|OPRK1|OPRM1 | opioid receptor agonist | Details | |
| C04773 | BRD-A45869167 | sal003 | EIF2A | eukaryotic translation initiation factor inhibitor | Details | |
| C04774 | BRD-K37747025 | sanazole | Details | |||
| C04775 | BRD-A64064900 | sangivamycin | DNA inhibitor | Details | ||
| C04776 | BRD-K66898851 | sanguinarium-chloride | CASP3 | apoptosis stimulant | Details | |
| C04777 | BRD-K99741577 | SANT-1 | SHH|SMO | smoothened receptor antagonist | Details | |
| C04778 | BRD-K35781423 | SANT-2 | SHH|SMO | smoothened receptor antagonist | Details | |
| C04779 | BRD-K36859431 | sapropterin | NOS3|PAH|TH|TPH1 | phenylalanine 4-hydroxylase stimulant | Details | |
| C04780 | BRD-K09963420 | saquinavir | CYP3A4 | HIV protease inhibitor | Details | |
| C04781 | BRD-K75308783 | SAR-245409 | MTOR|PIK3CG | PI3K inhibitor | Details | |
| C04782 | BRD-K19540840 | saracatinib | ABL1|LCK|SRC|YES1 | src inhibitor | Details | |
| C04783 | BRD-K08525451 | sarafloxacin | bacterial DNA gyrase inhibitor | Details | ||
| C04784 | BRD-K51263939 | sarcosine | SLC6A9 | Glycine transporter 1 inhibitor | Details | |
| C04785 | BRD-A92448440 | sari-59-801 | Details | |||
| C04786 | BRD-K79878800 | saroglitazar | PPARA|PPARG | PPAR receptor agonist | Details | |
| C04787 | BRD-A34358106 | sarpogrelate | HTR2A|HTR2B|HTR2C | serotonin receptor antagonist | Details | |
| C04788 | BRD-K38904395 | SAR131675 | FLT4 | VEGFR inhibitor | Details | |
| C04789 | BRD-K72868067 | SAR405 | PIK3C3 | PI3K inhibitor | Details | |
| C04790 | BRD-K86736469 | SAR405838 | MDM2 | MDM inhibitor | Details | |
| C04791 | BRD-K56912469 | SAR407899 | ROCK1 | rho associated kinase inhibitor | Details | |
| C04792 | BRD-K48892307 | sasapyrine | PTGS1|PTGS2 | NFkB pathway inhibitor | Details | |
| C04793 | BRD-M31395033 | satraplatin | DNA alkylating agent | Details | ||
| C04794 | BRD-K98028353 | savolitinib | MET | c-Met inhibitor | Details | |
| C04795 | BRD-A81513827 | saxagliptin | DPP4 | dipeptidyl peptidase inhibitor | Details | |
| C04796 | BRD-K77677632 | SB-200646 | HTR2B|HTR2C | serotonin receptor antagonist | Details | |
| C04797 | BRD-K54330070 | SB-202190 | AKT1|ALOX5|CHEK1|GSK3B|LCK|MAPK1|MAPK11|MAPK12|MAPK14|MAPK8|PRKCA|ROCK1|RPS6KB1|SGK1 | p38 MAPK inhibitor | Details | |
| C04798 | BRD-K27141178 | SB-203186 | HTR4 | serotonin receptor antagonist | Details | |
| C04799 | BRD-A37704979 | SB-203580 | AKT1|ALOX5|CHEK1|CYP2D6|CYP3A4|GAK|GSK3B|LCK|MAPK1|MAPK10|MAPK11|MAPK12|MAPK14|MAPK8|MAPK9|PRKCA|RAF1|RIPK2|ROCK1|RPS6KB1|SGK1|SRC|TNF | p38 MAPK inhibitor | Details | |
| C04800 | BRD-A22707317 | SB-205384 | GABRA3|GABRA5|GABRA6 | GABA receptor modulator | Details |