CMap Candidates
CMap (Connectivity Map) candidates are extracted from CLUE (CMap and LINCS Unified Environment), with detailed information, e.g., perturbagen time and dose, compound structure, targets, SMILES, mechanism of action. Two publicly available gene expression profiles of CKD are used to calculate individual connectivity scores and corresponding statistical significances for these candidates.
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6125 records.
| CMap ID | Pert ID | Compound Name | Targets | MoA | Compound Aliases | |
|---|---|---|---|---|---|---|
| C01501 | BRD-K48988407 | cytochlor | Details | |||
| C01502 | BRD-K87737963 | cyt387 | JAK1|JAK2|JAK3 | Details | ||
| C01503 | BRD-K79353516 | CY208-243 | CALY | dopamine receptor agonist | Details | |
| C01504 | BRD-K87021635 | CZC-54252 | LRRK2 | leucine rich repeat kinase inhibitor | Details | |
| C01505 | BRD-K01377300 | CZC24832 | PIK3CG | PI3K inhibitor | Details | |
| C01506 | BRD-M12328004 | C106 | Details | |||
| C01507 | BRD-K83914624 | C11-Acetate | ABAT|ACE|AKR1C3|CA2|CELA1|ESR2|FFAR2|FFAR3|HPRT1|LTA4H|MMP12|NOS1|NOS3|PLA2G1B|PTPN1|SOD1|TXN | Details | ||
| C01508 | BRD-K43167535 | C34 | TLR4 | toll-like receptor inhibitor | Details | |
| C01509 | BRD-K73383190 | C646 | EP300 | histone acetyltransferase inhibitor | Details | |
| C01510 | BRD-K74377520 | D-(+)-maltose | AMY2B|MGAM | Details | ||
| C01511 | BRD-K64636206 | D-alpha-tocopheryl-succinate | Details | |||
| C01512 | BRD-K04657451 | D-delta-Tocopherol | Details | |||
| C01513 | BRD-K20879694 | D-limonene | Details | |||
| C01514 | BRD-K00911807 | D-Phenylalanine | CCBL1|CRH|HCAR3 | enkephalinase inhibitor | Details | |
| C01515 | BRD-K71822263 | D-Serine | GLRA1|GRIN1|GRIN2A|GRIN2B|GRIN2C|GRIN2D|SERPINB3 | glutamate receptor agonist | Details | |
| C01516 | BRD-K09132007 | D-4476 | CSNK1A1|CSNK1D|TGFB1 | TGF beta receptor inhibitor | Details | |
| C01517 | BRD-K26997899 | D-64131 | TUBB | microtubule inhibitor | Details | |
| C01518 | BRD-K32372024 | D-7193 | Details | |||
| C01519 | BRD-K01080633 | DAA-1106 | TSPO | benzodiazepine receptor agonist | Details | |
| C01520 | BRD-K38168441 | dabigatran | F2 | thrombin inhibitor | Details | |
| C01521 | BRD-K57041787 | dabigatran-etexilate | F2 | thrombin inhibitor | Details | |
| C01522 | BRD-K09951645 | dabrafenib | BRAF|LIMK1|NEK11|RAF1|SIK1 | RAF inhibitor | Details | |
| C01523 | BRD-K35520305 | dacarbazine | PGD|POLA2 | DNA alkylating agent | Details | |
| C01524 | BRD-K56957086 | dacinostat | HDAC1|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 | HDAC inhibitor | Details | |
| C01525 | BRD-K82861010 | daclatasvir | HCV inhibitor | Details | ||
| C01526 | BRD-K57169635 | dacomitinib | EGFR|ERBB2|ERBB4 | EGFR inhibitor | Details | |
| C01527 | BRD-K70578146 | dactinomycin | POLR2A | RNA polymerase inhibitor | Details | |
| C01528 | BRD-K42095107 | daidzein | ESRRA|ESRRB|ESRRG|TRPC5 | estrogen receptor agonist | Details | |
| C01529 | BRD-A89196962 | dalargin | OPRM1 | opioid receptor agonist | Details | |
| C01530 | BRD-K30177383 | dalbavancin | PNLIP | bacterial cell wall synthesis inhibitor | Details | |
| C01531 | BRD-K18849474 | dalcetrapib | CETP | cholesteryl ester transfer protein inhibitor | Details | |
| C01532 | BRD-K22482860 | dalfampridine | KCNA1|KCNA10|KCNA2|KCNA3|KCNA4|KCNA5|KCNA6|KCNA7|KCNB1|KCNB2|KCNC1|KCNC2|KCNC3|KCNC4|KCND1|KCND2|KCND3|KCNF1|KCNG1|KCNG2|KCNG3|KCNG4|KCNH1|KCNH2|KCNH3|KCNH4|KCNH5|KCNH6|KCNH7|KCNH8|KCNJ13|KCNJ5|KCNQ1|KCNQ2|KCNQ3|KCNQ4|KCNQ5|KCNS1|KCNS2|KCNS3|KCNV1|KCNV2 | potassium channel blocker | Details | |
| C01533 | BRD-K26813177 | daltroban | TBXA2R | thromboxane receptor antagonist | Details | |
| C01534 | BRD-K83452553 | daminozide | KDM2A|KDM7A|PHF8 | KDM2A inhibitor | Details | |
| C01535 | BRD-A92537424 | danazol | AR|CCL2|ESR1|GNRHR|GNRHR2|PGR | estrogen receptor antagonist; progesterone receptor agonist | Details | |
| C01536 | BRD-K35589454 | danegaptide | gap junction modulator | Details | ||
| C01537 | BRD-K13769342 | danirixin | CXCR2 | CC chemokine receptor antagonist | Details | |
| C01538 | BRD-K45916615 | danofloxacin | bacterial DNA gyrase inhibitor | Details | ||
| C01539 | BRD-K08111240 | danoprevir | HCV inhibitor | Details | ||
| C01540 | BRD-K81272440 | dantrolene | RYR1|RYR3 | calcium channel blocker | Details | |
| C01541 | BRD-K10065684 | dantron | laxative | Details | ||
| C01542 | BRD-K07881437 | danusertib | AURKA|AURKB|AURKC|FGFR1|NTRK1|RET|SLK | Aurora kinase inhibitor; growth factor receptor inhibitor | Details | |
| C01543 | BRD-K58160573 | dapagliflozin | SLC5A1|SLC5A2 | sodium/glucose cotransporter inhibitor | Details | |
| C01544 | BRD-K61269089 | daphnetin | protein kinase inhibitor | Details | ||
| C01545 | BRD-K33133047 | dapiprazole | ADRA1A|ADRA1B|ADRA1D | adrenergic receptor antagonist | Details | |
| C01546 | BRD-K12885236 | dapivirine | CYP3A4|CYP3A5 | non-nucleoside reverse transcriptase inhibitor | Details | |
| C01547 | BRD-K51579475 | dapoxetine | HTR1A|HTR1B|HTR2C|SLC6A4 | selective serotonin reuptake inhibitor (SSRI) | Details | |
| C01548 | BRD-K06455935 | daprodustat | EGLN1 | hypoxia inducible factor inhibitor | Details | |
| C01549 | BRD-K62363391 | dapsone | DHFR | bacterial antifolate | Details | |
| C01550 | BRD-K47177710 | DAPT | gamma secretase inhibitor | Details | ||
| C01551 | BRD-K94358652 | daptomycin | bacterial cell wall synthesis inhibitor | Details | ||
| C01552 | BRD-K19085898 | darapladib | PLA2G7 | phospholipase inhibitor | Details | |
| C01553 | BRD-K82908348 | darglitazone | PPARG | PPAR receptor antagonist | Details | |
| C01554 | BRD-K95773607 | darifenacin | CHRM1|CHRM2|CHRM3|CHRM4|CHRM5 | acetylcholine receptor antagonist | Details | |
| C01555 | BRD-K84986517 | darunavir | CYP3A4 | HIV protease inhibitor | Details | |
| C01556 | BRD-K54863166 | darusentan | EDNRA | endothelin receptor antagonist | Details | |
| C01557 | BRD-K02943813 | dasabuvir | HCV inhibitor | Details | ||
| C01558 | BRD-K49328571 | dasatinib | ABL1|ABL2|BLK|EPHA2|FGR|FRK|FYN|HCK|KIT|LCK|LYN|PDGFRB|SRC|SRMS|STAT5B|YES1 | Bcr-Abl kinase inhibitor; ephrin inhibitor; KIT inhibitor; PDGFR tyrosine kinase receptor inhibitor; src inhibitor; tyrosine kinase inhibitor | Details | |
| C01559 | BRD-K31633810 | DAU-5884 | CHRM3 | acetylcholine receptor antagonist | Details | |
| C01560 | BRD-K14276241 | daucosterol | apoptosis stimulant | Details | ||
| C01561 | BRD-K43389675 | daunorubicin | TOP2A|TOP2B | RNA synthesis inhibitor; topoisomerase inhibitor | Details | |
| C01562 | BRD-K20738689 | dazmegrel | TBXAS1 | thromboxane synthase inhibitor | Details | |
| C01563 | BRD-K82767007 | dazoxiben | TBXAS1 | thromboxane synthase inhibitor | Details | |
| C01564 | BRD-K59204667 | DBeQ | CASP3 | ATPase inhibitor | Details | |
| C01565 | BRD-K83020231 | DBPR108 | DPP4 | dipeptidyl peptidase inhibitor | Details | |
| C01566 | BRD-K10596918 | DC-260126 | FFAR1 | free fatty acid receptor antagonist | Details | |
| C01567 | BRD-K49246350 | DCC-2618 | KIT|PDGFRA | PDGFR tyrosine kinase receptor inhibitor; KIT inhibitor | Details | |
| C01568 | BRD-K89299012 | DCEBIO | KCNN2|KCNN3|KCNN4 | potassium channel activator | Details | |
| C01569 | BRD-A39255369 | DCPIB | SLC1A2 | chloride channel blocker; gap junction modulator; glutamate inhibitor | Details | |
| C01570 | BRD-K61845293 | DDR1-IN-1 | DDR1|DDR2 | discoidin domain receptor inhibitor | Details | |
| C01571 | BRD-K80419150 | debrisoquin | SLC6A2 | adrenergic neuron blocker | Details | |
| C01572 | BRD-K49783248 | decamethonium | ACHE|CHRNA2 | acetylcholine receptor agonist | Details | |
| C01573 | BRD-A56320380 | decamethoxine | antiseptic | Details | ||
| C01574 | BRD-A95300432 | decernotinib | JAK3 | JAK inhibitor | Details | |
| C01575 | BRD-K79254416 | decitabine | DNMT1|DNMT3A | DNA methyltransferase inhibitor | Details | |
| C01576 | BRD-K17641316 | decoquinate | antiprotozoal agent | Details | ||
| C01577 | BRD-K43578482 | defactinib | PTK2 | focal adhesion kinase inhibitor | Details | |
| C01578 | BRD-K97010173 | deferasirox | CYP3A4 | chelating agent | Details | |
| C01579 | BRD-K06878038 | deferiprone | UGT1A6 | chelating agent | Details | |
| C01580 | BRD-K09821361 | deferoxamine-mesylate | chelating agent | Details | ||
| C01581 | BRD-K96006502 | deflazacort | NR3C1 | glucocorticoid receptor agonist | Details | |
| C01582 | BRD-K62304154 | deforolimus | MTOR | mTOR inhibitor | Details | |
| C01583 | BRD-A88562598 | degarelix | GNRHR | gonadotropin releasing factor hormone receptor antagonist | Details | |
| C01584 | BRD-A17300716 | dehydroacetic-acid | Details | |||
| C01585 | BRD-A64125466 | dehydrocholate | Details | |||
| C01586 | BRD-A11551002 | dehydrocholate-acid | Details | |||
| C01587 | BRD-K67186445 | dehydrocorydaline | ACHE | acetylcholinesterase inhibitor | Details | |
| C01588 | BRD-K41256143 | dehydroepiandrosterone | ESR1|ESR2|G6PD|GABRA1|GABRA2|GABRA3|GABRA4|GABRA5|GABRA6|GABRB1|GABRB2|GABRB3|GABRD|GABRE|GABRG1|GABRG2|GABRG3|GABRP|GABRQ|GRIN1|GRIN2A|GRIN2B|GRIN2C|GRIN2D|GRIN3A|GRIN3B|HSD17B1|NR1I2|NR1I3|PPARA|SIGMAR1|SULT2A1|SULT2B1 | protein synthesis stimulant | Details | |
| C01589 | BRD-K15360631 | dehydroepiandrosterone-sulfate | AR|ESR1|ESR2 | androgen receptor agonist; estrogen receptor agonist | Details | |
| C01590 | BRD-K17480742 | delamanid | bacterial cell wall synthesis inhibitor | Details | ||
| C01591 | BRD-K59325863 | delanzomib | CMA1|CTSG|CYP3A4|ELANE | proteasome inhibitor | Details | |
| C01592 | BRD-K00573984 | delapril | ACE | angiotensin converting enzyme inhibitor | Details | |
| C01593 | BRD-K34068325 | delavirdine | CYP3A4 | non-nucleoside reverse transcriptase inhibitor | Details | |
| C01594 | BRD-K45503887 | delivert | AGTR1|AGTR2 | angiotensin receptor agonist | Details | |
| C01595 | BRD-K79107392 | delphinidin | GLO1 | membrane permeability inhibitor | Details | |
| C01596 | BRD-K85776940 | delta-Tocotrienol | HMGCR | HMGCR inhibitor | Details | |
| C01597 | BRD-K90830492 | deltarasin | KRAS | phosphodiesterase inhibitor | Details | |
| C01598 | BRD-K51471001 | demecarium | ACHE|BCHE | acetylcholinesterase inhibitor | Details | |
| C01599 | BRD-A34145622 | demeclocycline | bacterial 30S ribosomal subunit inhibitor | Details | ||
| C01600 | BRD-K34122555 | denatonium-benzoate | Details |